James M. Balkovec: search on Z-Library

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1

The First Stereoselective Total Synthesis of Quinine

Niu, Deqiang, Fujimoto, A., Koft, Emil R., Balkovec, James M., Tata, James R., Dake, Gregory R., Stork, Gilbert

Journal:

Journal of the American Chemical Society

Year:

2001

Language:

english

File:

PDF, 120 KB

english, 2001

2

Novel orally active inhibitors of β-1,3-glucan synthesis derived from enfumafungin

Apgar, James M., Wilkening, Robert R., Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming Jo, Liberator,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.13 MB

english, 2015

3

Synthesis and Antifungal Activity of Novel Cationic Pneumocandin Bo Derivatives

Bouffard, F. Aileen, Zambias, Robert A., Dropinski, James F., Balkovec, James M., Hammond, Milton L., Abruzzo, George K., Bartizal, Kenneth F., Marrinan, Jean A., Kurtz, Myra B.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 520 KB

english, 1994

4

[Pharmacochemistry Library] Proceedings XIVth International Symposium on Medicinal Chemistry Volume 28 || The fungal cell wall as a drug discovery target: SAR of novel echinocandin analogs

Balkovec, James M.

Year:

1997

Language:

english

File:

PDF, 712 KB

english, 1997

5

Synthesis and structure-activity relationships of novel 3′-Hty-substituted pneumocandins

Regina M Black, James M Balkovec, Karl M Nollstadt, Sarah Dreikorn, Kenneth F Bartizal, George K Abruzzo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 361 KB

english, 1997

6

Synthesis and biological evaluation of antifungal derivatives of enfumafungin as orally bioavailable inhibitors of β-1,3-glucan synthase

Heasley, Brian H., Pacofsky, Gregory J., Mamai, Ahmed, Liu, Hao, Nelson, Kingsley, Coti, Ghjuvanni, Peel, Michael R., Balkovec, James M., Greenlee, Mark L., Liberator, Paul, Meng, Dongfang, Parker, Da

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 813 KB

english, 2012

7

A total synthesis of plumericin, allamcin and allamandin. Part 2. A biomimetic strategy

Trost, Barry M., Balkovec, James M., Mao, Michael K. T.

Journal:

Journal of the American Chemical Society

Year:

1986

Language:

english

File:

PDF, 1.40 MB

english, 1986

8

Reduction studies of antifungal echinocandin lipopeptides. One step conversion of echinocandin B to echinocandin C.

James M. Balkovec, Regina M. Black

Journal:

Tetrahedron Letters

Year:

1992

Language:

english

File:

PDF, 306 KB

english, 1992

9

Basic carbapenem analogs: Synthesis and in vitro activity of 1.BETA.-methyl-2-(pyridylmethylthio)-carbapenems.

BALKOVEC, JAMES M., SZYMONIFKA, MICHAEL J., HECK, JAMES V., RATCLIFFE, RONALD W.

Journal:

The Journal of Antibiotics

Year:

1991

Language:

english

File:

PDF, 326 KB

english, 1991

10

Synthesis of 4-methylene-1-cyclopentenes

Barry M. Trost, James M. Balkovec, Steven R. Angle

Journal:

Tetrahedron Letters

Year:

1986

Language:

english

File:

PDF, 184 KB

english, 1986

11

The total synthesis of allamandin

Barry M. Trost, James M. Balkovec

Journal:

Tetrahedron Letters

Year:

1985

Language:

english

File:

PDF, 173 KB

english, 1985

12

Synthesis, stability, and biological evaluation of water-soluble prodrugs of a new echinocandin lipopeptide. Discovery of a potential clinical agent for the treatment of systemic candidiasis and Pneumocystis carinii pneumonia (PCP)

Balkovec, James M., Black, Regina M., Hammond, Milton L., Heck, James V., Zambias, Robert A., Abruzzo, George, Bartizal, Ken, Kropp, Helmut, Trainor, Charlotte

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 718 KB

english, 1992

13

The First Stereoselective Total Synthesis of Quinine [ J. Am. Chem. Soc. 2001 , 123 (14), 3239−3242].

Stork, Gilbert, Niu, Deqiang, Fujimoto, Roger A., Koft, Emil R., Balkovec, James M., Tata, James R., Dake, Gregory R.

Journal:

Journal of the American Chemical Society

Year:

2001

Language:

english

File:

PDF, 38 KB

english, 2001

14

Novel N- Arylpyrazolo[3,2- c ]-Based Ligands for the Glucocorticoid Receptor: Receptor Binding and in Vivo Activity

Ali, Amjad, Thompson, Christopher F., Balkovec, James M., Graham, Donald W., Hammond, Milton L., Quraishi, Nazia, Tata, James R., Einstein, Monica, Ge, Lan, Harris, Georgianna, Kelly, Terri M., Mazur,

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 274 KB

english, 2004

15

Bicyclo[2.2.2]octyltriazole inhibitors of 11β-hydoxysteroid dehydrogenase type 1. Pharmacological agents for the treatment of metabolic syndrome

Milana Maletic, Aaron Leeman, Michael Szymonifka, Steven S. Mundt, Hratch J. Zokian, Kashmira Shah, Jasminka Dragovic, Kathy Lyons, Rolf Thieringer, Anne H. Vosatka, James Balkovec, Sherman T. Waddell

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 629 KB

english, 2011

16

Novel glucocorticoids containing a 6,5-bicyclic core fused to a pyrazole ring: Synthesis, in vitro profile, molecular modeling studies, and in vivo experiments

Christopher F. Thompson, Nazia Quraishi, Amjad Ali, Ralph T. Mosley, James R. Tata, Milton L. Hammond, James M. Balkovec, Monica Einstein, Lan Ge, Georgianna Harris, Terri M. Kelly, Paul Mazur, Shilpa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 331 KB

english, 2007

17

Inhibition of IMP-1 metallo-β-lactamase and sensitization of IMP-1-producing bacteria by thioester derivatives

Gail G. Hammond, Joann L. Huber, Mark L. Greenlee, Joanne B. Laub, Katherine Young, Lynn L. Silver, James M. Balkovec, KellyAnn D. Pryor, Joseph K. Wu, Barbara Leiting, David L. Pompliano, Jeffrey H.

Journal:

FEMS Microbiology Letters

Year:

1999

Language:

english

File:

PDF, 319 KB

english, 1999

18

4-Methyl-5-phenyl triazoles as selective inhibitors of 11β-hydroxysteroid dehydrogenase type I

Yuping Zhu, Steven H. Olson, Anne Hermanowski-Vosatka, Steven Mundt, Kashmira Shah, Marty Springer, Rolf Thieringer, Samuel Wright, Jianying Xiao, Hratch Zokian, James M. Balkovec

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 294 KB

english, 2008

19

Synthesis of oxaspiropiperidines as a strategy for lowering log D

Timothy Cernak, Kevin Dykstra, Dorothy Levorse, Andreas Verras, James Balkovec, Ravi Nargund, Robert DeVita

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 612 KB

english, 2011

20

[Annual Reports in Medicinal Chemistry] Volume 33 || Non-Azole Antifungal Agents

Balkovec, James M.

Year:

1998

Language:

english

File:

PDF, 753 KB

english, 1998

21

Substituted phenyl triazoles as selective inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1

Wanying Sun, Milana Maletic, Steven S. Mundt, Kashmira Shah, Hratch Zokian, Kathy Lyons, Sherman T. Waddell, James Balkovec

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 676 KB

english, 2011

22

Inhibition of IMP-1 metallo-β-lactamase and sensitization of IMP-1-producing bacteria by thioester derivatives

Gail G. Hammond, Joann L. Huber, Mark L. Greenlee, Joanne B. Laub, Katherine Young, Lynn L. Silver, James M. Balkovec, KellyAnn D. Pryor, Joseph K. Wu, Barbara Leiting, David L. Pompliano, Jeffrey H.

Journal:

FEMS Microbiology Letters

Year:

1999

Language:

english

File:

PDF, 316 KB

english, 1999

23

The First Stereoselective Total Synthesis of Quinine.

Gilbert Stork, Deqiang Niu, A. Fujimoto, Emil R. Koft, James M. Balkovec, James R. Tata, Gregory R. Dake

Journal:

Year:

2001

File:

PDF, 23 KB

2001

24

Pneumocandin antifungal lipopeptides. The phenolic hydroxyl is required for 1,3-β-glucan synthesis inhibition.

James M. Balkovec, Regina M. Black, George K. Abruzzo, Ken Bartizal, Sarah Dreikorn, Nollstadt Karl

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 306 KB

english, 1993

25

Preclinical Evaluation of the Stability, Safety, and Efficacy of CD101, a Novel Echinocandin

Ong, Voon, Hough, Grayson, Schlosser, Michael, Bartizal, Ken, Balkovec, James M., James, Kenneth D., Krishnan, B. Radha

Journal:

Antimicrobial Agents and Chemotherapy

Year:

2016

Language:

english

File:

PDF, 1.11 MB

english, 2016

26

Efficacy of MK-991 (L-743,872), a Semisynthetic Pneumocandin, in Murine Models ofPneumocystis carinii

Powles, Mary Ann, Liberator, Paul, Anderson, Jennifer, Karkhanis, Yashwant, Dropinski, James F., Bouffard, F. Aileen, Balkovec, James M., Fujioka, Hisashi, Aikawa, Masamichi, McFadden, Diane, Schmatz,

Journal:

Antimicrobial Agents and Chemotherapy

Year:

1998

File:

PDF, 1.06 MB

1998

27

A biomimetic approach to plumericin

Trost, Barry M., Balkovec, James M., Mao, Michael K. T.

Journal:

Journal of the American Chemical Society

Year:

1983

Language:

english

File:

PDF, 397 KB

english, 1983

28

Antifungal lipopeptides: Structure-activity relationships of 3-hydroxyglutamine-modified pneumocandin B0 derivatives

Robert A. Zambias, Catherine James, Milton L. Hammond, George K. Abruzzo, Kenneth F. Bartizal, Karl H. Nollstadt, Cameron Douglas, Jean Marrinan, James M. Balkovec

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 326 KB

english, 1995

29

On the use of the O-methylmandelate ester for establishment of absolute configuration of secondary alcohols

Trost, Barry M., Belletire, John L., Godleski, Stephen, McDougal, Patrick G., Balkovec, James M., Baldwin, John J., Christy, Marcia E., Ponticello, Gerald S., Varga, Sandor L., Springer, James P.

Journal:

Journal of Organic Chemistry

Year:

1986

Language:

english

File:

PDF, 593 KB

english, 1986

30

Ibrexafungerp: an orally active Î²-1,3-glucan synthesis inhibitor

Apgar, James M., Wilkening, Robert R., Parker, Dann L., Meng, Dongfang, Wildonger, Kenneth J., Sperbeck, Donald, Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, A

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 462 KB

2020

31

Determination of the Absolute Stereochemistry of (−)-Galbonolide A

Tse, Bruno, Blazey, Charles M., Tu, Ben, Balkovec, James

Journal:

Journal of Organic Chemistry

Year:

1997

Language:

english

File:

PDF, 186 KB

english, 1997

32

Novel ketal ligands for the glucocorticoid receptor: in vitro and in vivo activity

Cameron J. Smith, Amjad Ali, James M. Balkovec, Donald W. Graham, Milton L. Hammond, Gool F. Patel, Gregory P. Rouen, Scott K. Smith, James R. Tata, Monica Einstein, Lan Ge, Georgianna S. Harris, Ther

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 234 KB

english, 2005

33

Lipopeptide antifungal agents: Amine conjugates of the semi-synthetic pneumocandins L-731,373 and L-733,560

Robert A. Zambias, Catherine James, George K. Abruzzo, Kenneth F. Bartizal, Richard Hajdu, Randy Thompson, Karl H. Nollstadt, Jean Marrinan, James M. Balkovec

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 353 KB

english, 1997

34

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Christopher F. Thompson, Nazia Quraishi, Amjad Ali, James R. Tata, Milton L. Hammond, James M. Balkovec, Monica Einstein, Lan Ge, Georgianna Harris, Theresa M. Kelly, Paul Mazur, Shilpa Pandit, Joseph

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 127 KB

english, 2005

35

Synthesis and SAR of thioester and thiol inhibitors of IMP-1 Metallo-β-Lactamase

Mark L. Greenlee, Joanne B. Laub, James M. Balkovec, Milton L. Hammond, Gail G. Hammond, David L. Pompliano, Jeffrey H. Epstein-Toney

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 408 KB

english, 1999

36

Alkyl side-chain derivatives of sordaricin as potent antifungal agents against yeast

Bruno Tse, James M. Balkovec, Charles M. Blazey, Ming-Jo Hsu, Jennifer Nielsen, Dennis Schmatz

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 213 KB

english, 1998

37

A total synthesis of plumericin, allamcin, and allamandin. Part 1. Basic strategy

Trost, Barry M., Mao, Michael K. T., Balkovec, James M., Buhlmayer, Peter.

Journal:

Journal of the American Chemical Society

Year:

1986

Language:

english

File:

PDF, 1.19 MB

english, 1986

38

Section Review: Anti-infectives: Lipopeptide antifungal agents

Balkovec, James M

Journal:

Expert Opinion on Investigational Drugs

Year:

1994

Language:

english

File:

PDF, 1.88 MB

english, 1994

39

MK-5204: an orally active Î²-1,3-glucan synthesis inhibitor

Apgar, James M., Wilkening, Robert R., Parker, Dann L., Meng, Dongfang, Wildonger, Kenneth J., Sperbeck, Donald, Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, A

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2020

File:

PDF, 451 KB

2020

40

Discovery of betamethasone 17α-carbamates as dissociated glucocorticoid receptor modulators in the rat

Amjad Ali, James M. Balkovec, Mark Greenlee, Milton L. Hammond, Greg Rouen, Gayle Taylor, Monica Einstein, Lan Ge, Georgianna Harris, Terri M. Kelly, Paul Mazur, Shilpa Pandit, Joseph Santoro, Ayesha

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 263 KB

english, 2008

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